Small Molecule Inhibitors of Zinc-dependent Histone Deacetylases
- 1 October 2013
- journal article
- review article
- Published by Elsevier BV in Neurotherapeutics
- Vol. 10 (4), 589-604
- https://doi.org/10.1007/s13311-013-0226-1
Abstract
No abstract availableKeywords
This publication has 100 references indexed in Scilit:
- Class I HDACs Share a Common Mechanism of Regulation by Inositol PhosphatesMolecular Cell, 2013
- Histone deacetylase modulators provided by Mother NatureGenes & Nutrition, 2012
- Discovery of histone deacetylase 8 selective inhibitorsBioorganic & Medicinal Chemistry Letters, 2011
- On the inhibition of histone deacetylase 8Bioorganic & Medicinal Chemistry, 2010
- Multiple roles of HDAC inhibition in neurodegenerative conditionsTrends in Neurosciences, 2009
- Histone Deacetylase Inhibitor MS-275 Exhibits Poor Brain Penetration: Pharmacokinetic Studies of [11C]MS-275 using Positron Emission TomographyACS Chemical Neuroscience, 2009
- Molecular modifications on carboxylic acid derivatives as potent histone deacetylase inhibitors: Activity and docking studiesBioorganic & Medicinal Chemistry, 2009
- Searching for Disease Modifiers—PKC Activation and HDAC Inhibition—A Dual Drug Approach to Alzheimer's Disease that Decreases Aβ Production while Blocking Oxidative StressChemMedChem, 2009
- Structural Studies of Human Histone Deacetylase 8 and Its Site-Specific Variants Complexed with Substrate and Inhibitors,Biochemistry, 2008
- Epigenetic targets of HDAC inhibition in neurodegenerative and psychiatric disordersCurrent Opinion in Pharmacology, 2008