Efficient synthesis of piperazine-2,6-dione and 4-(1H-indole-2-carbonyl)piperazine-2,6-dione derivatives and their evaluation for anticancer activity
- 16 January 2013
- journal article
- Published by Springer Science and Business Media LLC in Medicinal Chemistry Research
- Vol. 22 (10), 4600-4609
- https://doi.org/10.1007/s00044-012-0438-7
Abstract
No abstract availableKeywords
This publication has 25 references indexed in Scilit:
- A Mouse Model for Studying the Interaction of Bisdioxopiperazines with Topoisomerase IIα in VivoMolecular Pharmacology, 2007
- Synthesis of Symmetrically 1,4-disubstituted piperazine-2,5-diones: A New Class of Antileishmanial AgentsJournal of Chemical Research, 2007
- Controlling Pathogenic Gram-Negative Bacteria by Interfering with Their Biofilm FormationDrug Design Reviews - Online, 2005
- Structure-Based Exploration of Cyclic Dipeptide Chitinase InhibitorsJournal of Medicinal Chemistry, 2004
- Synthesis of Diketopiperazines Containing Prolinyl Unit — Cyclo(L-prolinyl-L-leucine), Cyclo(L-prolinyl-L-isoleucine) and Cyclo(L-tryptophyl-L-proline).ChemInform, 2004
- Synthesis and in vitro evaluation of a series of diketopiperazine inhibitors of plasminogen activator inhibitor-1Bioorganic & Medicinal Chemistry Letters, 2001
- A new class of highly cytotoxic diketopiperazinesBioorganic & Medicinal Chemistry Letters, 2000
- Solution-phase combinatorial synthesis and evaluation of piperazine-2,5-dione derivativesBioorganic & Medicinal Chemistry Letters, 2000
- The design of potent and selective inhibitors of thrombin utilizing a piperazinedione template: Part 2Bioorganic & Medicinal Chemistry Letters, 1999
- Inhibition of Plasminogen Activator Inhibitor-1 Activity by Two Diketopiperazines, XR330 and XR334 Produced by Streptomyces sp.The Journal of Antibiotics, 1996