Synthesis of a novel benzyl-octahydropyrazino[1,2-a]pyrimidin-6-one derivative as a convenient internal bicyclic peptidomimetic
- 31 March 2008
- journal article
- research article
- Published by Elsevier BV in Tetrahedron Letters
- Vol. 49 (14), 2316-2319
- https://doi.org/10.1016/j.tetlet.2008.01.137
Abstract
No abstract availableKeywords
This publication has 21 references indexed in Scilit:
- Synthesis of constrained analogues of cholecystokinin/opioid chimeric peptidesTetrahedron Letters, 2006
- An Anomeric Control on Remote Stereochemistry in the Synthesis of SpiroketalsJournal of the American Chemical Society, 2005
- Parallel synthesis and biological evaluation of different sizes of bicyclo[2,3]‐Leu‐enkephalin analoguesPeptide Science, 2005
- Cyclizations of N-Acyliminium IonsChemical Reviews, 2004
- Design, Synthesis, and Evaluation of Opioid Analogues with Non-Peptidic β-Turn Scaffold: Enkephalin and Endomorphin MimeticsJournal of Medicinal Chemistry, 2002
- Solid-Phase Syntheses of β-Turn Analogues To Mimic or Disrupt Protein−Protein InteractionsAccounts of Chemical Research, 2001
- Design and Synthesis of Novel Conformationally Restricted Peptide Secondary Structure MimeticsOrganic Letters, 2000
- Solid-Phase Synthesis and Structural Analysis of Bicyclic β-Turn Mimetics Incorporating Functionality at theitoi+ 3 PositionsJournal of the American Chemical Society, 1999
- Harmonic Vibrational Frequencies: An Evaluation of Hartree−Fock, Møller−Plesset, Quadratic Configuration Interaction, Density Functional Theory, and Semiempirical Scale FactorsThe Journal of Physical Chemistry, 1996
- Synthesis of a bicyclic γ-lactam dipeptide analogueTetrahedron Letters, 1993