Design and Synthesis of Novel Conformationally Restricted Peptide Secondary Structure Mimetics
- 11 January 2000
- journal article
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 2 (3), 301-302
- https://doi.org/10.1021/ol990355r
Abstract
[structure: see text] A facile synthesis of the novel conformationally restricted reverse turn mimetic is described. The key features are the preparation of the alpha-keto amide and tandem bicyclic ring formation.Keywords
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