An Improved Procedure for the Synthesis of Nucleoside Phosphoramidates
- 12 September 2002
- journal article
- research article
- Published by American Chemical Society (ACS) in Organic Process Research & Development
- Vol. 6 (6), 819-822
- https://doi.org/10.1021/op025562c
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- Synthesis and Antiviral Evaluation of Phosphoramidate Derivatives of (E)-5-(2-Bromovinyl)-2′-DeoxyuridineAntiviral Chemistry and Chemotherapy, 2001
- A Novel Approach to Thymidylate Synthase as a Target for Cancer ChemotherapyMolecular Pharmacology, 2001
- Synthesis of a phosphoramidate pro-drug of 6-thio-7-deaza-2′-deoxyguanosine (TDG): a regioselective phosphorylationTetrahedron Letters, 2001
- 5‘-Phosphoramidates and 5‘-Diphosphates of 2‘-O-Allyl-β-d-arabinofuranosyl- uracil, -cytosine, and -adenine: Inhibition of Ribonucleotide ReductaseJournal of Medicinal Chemistry, 1999
- The Presence of Substituents on the Aryl Moiety of the Aryl Phosphoramidate Derivative of d4T Enhances Anti-HIV Efficacy in Cell Culture: A Structure−Activity RelationshipJournal of Medicinal Chemistry, 1999
- Certain phosphoramidate derivatives of dideoxy uridine (ddU) are active against HIV and successfully by-pass thymidine kinaseFEBS Letters, 1994
- N?-Phosphoarginine Phosphatase from Rat Renal Microsome Was Alkaline PhosphataseArchives of Biochemistry and Biophysics, 1994
- Aryl phosphate derivatives of AZT retain activity against HIV1 in cell lines which are resistant to the action of AZTAntiviral Research, 1992
- The synthesis of the potent anti-herpes virus agent, E-5(2-bromovinyl)-2′-deoxyuridine and related compoundsTetrahedron Letters, 1979
- Metabolism of phosphoramidates I. Enzymic hydrolysis and transfer reactionsBiochimica et Biophysica Acta, 1962