Synthesis and Evaluation of α-Thymidine Analogues as Novel Antimalarials
Open Access
- 14 December 2012
- journal article
- research article
- Published by American Chemical Society (ACS) in Journal of Medicinal Chemistry
- Vol. 55 (24), 10948-10957
- https://doi.org/10.1021/jm301328h
Abstract
No abstract availableKeywords
This publication has 28 references indexed in Scilit:
- European Vaccine Initiative: lessons from developing malaria vaccinesExpert Review of Vaccines, 2011
- Exploring new inhibitors of Plasmodium falciparum purine nucleoside phosphorylaseEuropean Journal of Medicinal Chemistry, 2010
- Potential application of thymidylate kinase in nucleoside analogue activation in Plasmodium falciparumBioorganic & Medicinal Chemistry, 2010
- Novel Inhibitors of Plasmodium falciparum Dihydroorotate Dehydrogenase with Anti-malarial Activity in the Mouse Model*Published by Elsevier BV ,2010
- Malaria: a research agenda for the eradication eraThe Lancet, 2009
- Mutational, inhibitory and microcalorimetric analyses of Plasmodium falciparum TMP kinase. Implications for drug discoveryParasitology, 2009
- Targeting DHFR in parasitic protozoaDrug Discovery Today, 2005
- Genome sequence of the human malaria parasite Plasmodium falciparumNature, 2002
- Drugs to Combat Tropical Protozoan ParasitesScience, 2002
- Enzymes of purine and pyrimidine metabolism from the human malaria parasite, Plasmodium falciparumMolecular and Biochemical Parasitology, 1982