Cefiderocol (S-649266), A new siderophore cephalosporin exhibiting potent activities against Pseudomonas aeruginosa and other gram-negative pathogens including multi-drug resistant bacteria: Structure activity relationship
- 1 July 2018
- journal article
- research article
- Published by Elsevier BV in European Journal of Medicinal Chemistry
- Vol. 155, 847-868
- https://doi.org/10.1016/j.ejmech.2018.06.014
Abstract
No abstract availableKeywords
This publication has 39 references indexed in Scilit:
- Preparation, Gram-Negative Antibacterial Activity, and Hydrolytic Stability of Novel Siderophore-Conjugated Monocarbam DiolsACS Medicinal Chemistry Letters, 2011
- Design, synthesis, and structure–activity relationship study of bicyclic piperazine analogs of indole-3-carboxamides as novel cannabinoid CB1 receptor agonistsBioorganic & Medicinal Chemistry Letters, 2010
- Chemistry and biology of siderophoresNatural Product Reports, 2010
- Multidrug-Resistant Gram-Negative InfectionsDrugs, 2009
- Synthesis and SAR of novel parenteral anti-pseudomonal cephalosporins: Discovery of FR264205Bioorganic & Medicinal Chemistry Letters, 2008
- A novel series of parenteral cephalosporins exhibiting potent activities against both Pseudomonas aeruginosa and other Gram-negative pathogens. Part 2: Synthesis and structure–activity relationshipsBioorganic & Medicinal Chemistry, 2008
- DPPH (= 2,2‐Diphenyl‐1‐picrylhydrazyl = 2,2‐Diphenyl‐1‐(2,4,6‐trinitrophenyl)hydrazyl) Radical‐Scavenging Reaction of Protocatechuic Acid Esters (= 3,4‐Dihydroxybenzoates) in Alcohols: Formation of Bis‐alcohol AdductHelvetica Chimica Acta, 2006
- Enterobactin: the characteristic catecholate siderophore of Enterobacteriaceae is produced byStreptomycesspeciesFEMS Microbiology Letters, 2001
- Synthesis and biological activity of a novel class of cephalosporins with a oxadiazolyl hydroxypyridone moiety at C-7Bioorganic & Medicinal Chemistry Letters, 1995
- Synthesis, renal vasodilator and dopamine‐sensitive adenylate cyclase activities of O‐Methyl derivatives of 6‐chloro‐2,3,4,5‐tetr ahydro‐1‐(4‐hydroxyphenyl)‐1H‐3‐benzazepin‐7,8‐diol (SK&F 82526)Journal of Heterocyclic Chemistry, 1986