Receptor-specific functional efficacies of alkyl imidazoles as dual histamine H3/H4 receptor ligands
- 11 March 2011
- journal article
- Published by Elsevier BV in European Journal of Pharmacology
- Vol. 654 (3), 200-208
- https://doi.org/10.1016/j.ejphar.2010.12.033
Abstract
No abstract availableKeywords
This publication has 36 references indexed in Scilit:
- In Silico Characterization of Ligand Binding Modes in the Human Histamine H4 Receptor and their Impact on Receptor ActivationChemBioChem, 2010
- H3 Histamine Receptor–Mediated Activation of Protein Kinase Cα Inhibits the Growth of Cholangiocarcinoma In vitro and In vivoMolecular Cancer Research, 2009
- Homology Model Adjustment and Ligand Screening with a Pseudoreceptor of the Human Histamine H4 ReceptorChemMedChem, 2009
- The histamine H4 receptor is functionally expressed on neurons in the mammalian CNSBritish Journal of Pharmacology, 2009
- Autoregulation of McA-RH7777 Hepatoma Cell Proliferation by Histamine H3ReceptorsThe Journal of pharmacology and experimental therapeutics, 2008
- Keynote review: Histamine H3 receptor antagonists reach out for the clinicDrug Discovery Today, 2005
- Distinct pharmacology of rat and human histamine H3 receptors: role of two amino acids in the third transmembrane domainBritish Journal of Pharmacology, 2000
- Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in LeukocytesPublished by Elsevier BV ,2000
- A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye bindingAnalytical Biochemistry, 1976
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973