Asymmetric synthesis and preliminary evaluation of (R)- and (S)-[11C]bisoprolol, a putative β1-selective adrenoceptor radioligand
- 28 February 2001
- journal article
- Published by Elsevier BV in Neurochemistry International
- Vol. 38 (2), 169-180
- https://doi.org/10.1016/s0197-0186(00)00049-8
Abstract
No abstract availableKeywords
This publication has 32 references indexed in Scilit:
- Pharmacokinetics of β‐adrenoceptor blockers in obese and normal volunteersBritish Journal of Clinical Pharmacology, 1997
- Stereoselective Pharmacokinetics of Bisoprolol After Intravenous and Oral Administration in Beagle DogsJournal of Pharmaceutical Sciences, 1997
- Lack of pineal β-adrenergic receptor alterations in suicide victims with major depressionPsychoneuroendocrinology, 1997
- Dose Proportionality of Bisoprolol Enantiomers in Humans After Oral Administration of the RacemateThe Journal of Clinical Pharmacology, 1994
- Synthesis and evaluation of 1′-[18F]fluorometoprolol as a potential tracer for the visualization of β-adrenoceptors with PETNuclear Medicine and Biology, 1993
- Preparation and in vivo binding of [11C]carazolol, a radiotracer for the beta-adrenergic receptorInternational Journal of Radiation Applications and Instrumentation. Part B. Nuclear Medicine and Biology, 1992
- Distribution of beta‐adrenergic receptor subtypes in human post‐mortem brain: Alterations in limbic regions of schizophrenicsSynapse, 1992
- Specific non- -adrenergic binding sites for 125I-iodocyanopindolol in myocardial membrane preparations: a comparative study between human, rat, and porcine heartsCardiovascular Research, 1991
- β-Adrenoceptor-Binding Studies of the Cardioselective β Blockers Bisoprolol, H-I 42 BS, and HX-CH 44 BS to Heart Membranes and Intact Ventricular Myocytes of Adult RatsJournal of Cardiovascular Pharmacology, 1990
- Synthesis of the 11C-labelled β-adrenergic receptor ligands atenolol, metoprolol and propranololInternational Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1989