Design, synthesis and bioassays of antagonists of LHRH which have high antiovulatory activity and release negligible histamine
- 26 October 1987
- journal article
- research article
- Published by Elsevier BV in Biochemical and Biophysical Research Communications
- Vol. 148 (2), 849-856
- https://doi.org/10.1016/0006-291x(87)90953-3
Abstract
No abstract availableThis publication has 9 references indexed in Scilit:
- Effect of reductive alkylation of D-lysine in position 6 on the histamine-releasing activity of luteinizing hormone-releasing hormone antagonistsJournal of Medicinal Chemistry, 1987
- New effective gonadotropin releasing hormone antagonists with minimal potency for histamine release in vitroJournal of Medicinal Chemistry, 1986
- Increased potency of antagonists of the luteinizing hormone releasing hormone which have D-3-Pal in position 6Biochemical and Biophysical Research Communications, 1986
- Gonadotropin-Releasing Hormone Analog Design. Structure-Function Studies Toward the Development of Agonists and Antagonists: Rationale and PerspectiveEndocrine Reviews, 1986
- Antagonists of the luteinizing hormone releasing hormone (LHRH) with emphasis on the Trp7 of the salmon and chicken II LHRH'sBiochemical and Biophysical Research Communications, 1984
- Luteinizing hormone-releasing hormone antagonists containing very hydrophobic amino acidsJournal of Medicinal Chemistry, 1984
- Synthesis and biological activity of LH-RH antagonists modified in position 1Peptides, 1982
- The effects of substance P on histamine and 5‐hydroxytryptamine release in the ratThe Journal of Physiology, 1982
- Peptide hormones. 109. Inhibitory analogs of the luteinizing hormone-releasing hormone having D-aromatic residues in positions 2 and 6 and variation in position 3Journal of Medicinal Chemistry, 1978