Favourable involvement of α2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancement
- 1 April 2012
- journal article
- Published by Elsevier BV in Bioorganic & Medicinal Chemistry
- Vol. 20 (7), 2259-2265
- https://doi.org/10.1016/j.bmc.2012.02.016
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Properly substituted 1,4-dioxane nucleus favours the selective M3 muscarinic receptor activationBioorganic & Medicinal Chemistry, 2009
- Structure−Activity Relationships in 1,4-Benzodioxan-Related Compounds. 9. From 1,4-Benzodioxane to 1,4-Dioxane Ring as a Promising Template of Novel α1D-Adrenoreceptor Antagonists, 5-HT1A Full Agonists, and Cytotoxic AgentsJournal of Medicinal Chemistry, 2008
- Novel Ligands Rationally Designed for Characterizing I2−Imidazoline Binding Sites Nature and FunctionsJournal of Medicinal Chemistry, 2008
- α2-Adrenoreceptors Profile Modulation. 4. From Antagonist to Agonist BehaviorJournal of Medicinal Chemistry, 2008
- Interest of α2-Adrenergic Agonists and Antagonists in Clinical Practice: Background, Facts and PerspectivesCurrent Topics in Medicinal Chemistry, 2007
- The analgesic efficacy of partial opioid agonists is increased in mice with targeted inactivation of the α2A-adrenoceptor geneEuropean Journal of Pharmacology, 2006
- Stimulation frequency-noradrenaline release relationships examined in α2A-, α2B- and α2C-adrenoceptor-deficient miceNaunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 2001
- Adrenoceptor subclassification: an approach to improved cardiovascular therapeuticsPharmaceutica Acta Helvetiae, 2000
- Separation of α-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazolineBioorganic & Medicinal Chemistry, 1995
- Epidural clonidine analgesia for intractable cancer painPain, 1995