Chemical and enzymatic oxidative coupling of 5-hydroxy-N-dimethyltryptamine with amines
- 1 July 1987
- journal article
- research article
- Published by American Chemical Society (ACS) in Journal of Medicinal Chemistry
- Vol. 30 (7), 1239-1241
- https://doi.org/10.1021/jm00390a020
Abstract
As part of a program aiming to obtain a covalent labeling of serotoninergic receptors we have studied the oxidative coupling of serotonin derivatives with amino compounds. The oxidation of bufotenine (2) by MnO2 and human ceruloplasmin followed by the Michael type addition with dansylcadaverine and dansyllysine gave a fluorescent adduct identified as fused oxazole structure 4.This publication has 11 references indexed in Scilit:
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