Polymer-supported chiral sulfonamide catalyzed one-pot reduction of β-keto nitriles: a practical synthesis of (R)-fluoxetine and (R)-duloxetine
- 1 May 2005
- journal article
- Published by Elsevier BV in Tetrahedron: Asymmetry
- Vol. 16 (10), 1873-1879
- https://doi.org/10.1016/j.tetasy.2005.04.002
Abstract
No abstract availableKeywords
This publication has 35 references indexed in Scilit:
- Enantioselective Reduction of Ketones Catalyzed by Polymer-Supported Sulfonamide Using NaBH4/Me3SiCl (or BF3⋅OEt2) as Reducing AgentAngewandte Chemie-International Edition, 2001
- Asymmetric Borane Reduction of Prochiral Ketones by Polymer-Supported Chiral SulfonamidesThe Journal of Organic Chemistry, 2000
- Enantioselective Reduction of Oxime Ethers with Borane Catalyzed by Polymer-Supported 2-PiperazinemethanolThe Journal of Organic Chemistry, 2000
- Asymmetric Hydrogenation of α, β, and γ-Aminoketones Catalyzed by Cationic Rhodium(I){AMPP} ComplexesSynlett, 1997
- Prozac (fluoxetine, lilly 110140), the first selective serotonin uptake inhibitor and an antidepressant drug: Twenty years since its first publicationLife Sciences, 1995
- Practical Asymmetric Synthesis of (R)-Fluoxetine Hydrochloride Catalyzed by (2S, 4S)-4-Dicyclohexylphosphino-2-diphenylphosphinomethyl-1-(N-methylcarbamoyl)pyrrolidine-Rhodium Complex1Synlett, 1991
- LY227942, an inhibitor of serotonin and norepinephrine uptake: Biochemical pharmacology of a potential antidepressant drugLife Sciences, 1988
- The absolute configurations and pharmacological activities of the optical isomers of fluoxetine, a selective serotonin-uptake inhibitorJournal of Medicinal Chemistry, 1988
- Molecular structure of fluoxetine hydrochloride, a highly selective serotonin-uptake inhibitorJournal of Medicinal Chemistry, 1988
- Asymmetric synthesis using chirally modified borohydrides. Part 2. Enantioselective reduction of ketones with polymeric (S)-prolinol–borane reagentJournal of the Chemical Society, Perkin Transactions 1, 1984