CuBr for KA2 reaction: en route to propargylic amines bearing a quaternary carbon center
- 1 August 2013
- journal article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- Vol. 49 (79), 8976-8978
- https://doi.org/10.1039/c3cc45301d
Abstract
A highly efficient CuBr-catalyzed coupling of ketones, amines and alkynes (KA2) forming propargylic amines bearing a quaternary carbon center with the broadest scope so far has been developed.Keywords
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