A novel photoaffinity label for the dopamine transporter based on N-substituted 3α-[bis(4′-fluorophenyl)methoxy]tropane
Open Access
- 2 December 1997
- journal article
- Published by Elsevier BV in Bioorganic & Medicinal Chemistry Letters
- Vol. 7 (23), 3027-3032
- https://doi.org/10.1016/s0960-894x(97)10139-1
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- 3‘-Chloro-3α-(diphenylmethoxy)tropane But Not 4‘-Chloro-3α- (diphenylmethoxy)tropane Produces a Cocaine-like Behavioral ProfileJournal of Medicinal Chemistry, 1997
- Dopamine Transporter Ligand Binding DomainsOnline Journal of Public Health Informatics, 1996
- 2-Carbomethoxy-3-(diarylmethoxy)-1αH,5αH-tropane Analogs: Synthesis and Inhibition of Binding at the Dopamine Transporter and Comparison with Piperazines of the GBR SeriesJournal of Medicinal Chemistry, 1996
- Novel 4'-Substituted and 4',4''-Disubstituted 3.alpha.-(Diphenylmethoxy)tropane Analogs as Potent and Selective Dopamine Uptake InhibitorsJournal of Medicinal Chemistry, 1995
- Novel 3.alpha.-(Diphenylmethoxy)tropane Analogs: Potent Dopamine Uptake Inhibitors without Cocaine-like Behavioral ProfilesJournal of Medicinal Chemistry, 1994
- Stereochemical requirements for pseudoirreversible inhibition of opioid mu receptor binding by the 3‐methylfentanyl congeners, RTI‐46144 and its enantiomers: Evidence for different binding domainsSynapse, 1993
- Radiosynthesis of a photoaffinity probe for the cocaine receptor of the dopamine transporter: 3β-(p-chlorophenyl)tropan-2β-carboxylic acid m-([125I]-iodo)-p-azidophenethyl ester ([125I]-RTI-82)Journal of Labelled Compounds and Radiopharmaceuticals, 1993
- Probes for the cocaine receptor. Potentially irreversible ligands for the dopamine transporterJournal of Medicinal Chemistry, 1992
- (+)-Cis-3-methylfentanyl and its analogs bind pseudoirreversibly to the mu opioid binding site: Evidence for pseudoallosteric modulationNeuropharmacology, 1991
- A one-pot radiosynthesis of [125I]iodoazido photoaffinity labelsJournal of Labelled Compounds and Radiopharmaceuticals, 1989