Identification of small molecule estrogen‐related receptor α–specific antagonists and homology modeling to predict the molecular determinants as the basis for selectivity over ERRβ and ERRγ
- 1 June 2008
- journal article
- research article
- Published by Wiley in Drug Development Research
- Vol. 69 (4), 203-218
- https://doi.org/10.1002/ddr.20246
Abstract
No abstract availableKeywords
This publication has 44 references indexed in Scilit:
- Structure-guided synthesis of tamoxifen analogs with improved selectivity for the orphan ERRγBioorganic & Medicinal Chemistry Letters, 2006
- Identification of a Selective Inverse Agonist for the Orphan Nuclear Receptor Estrogen-Related Receptor αJournal of Medicinal Chemistry, 2004
- Announcing the worldwide Protein Data BankNature Structural & Molecular Biology, 2003
- The SWISS-PROT protein knowledgebase and its supplement TrEMBL in 2003Nucleic Acids Research, 2003
- 4-Hydroxytamoxifen binds to and deactivates the estrogen-related receptor γProceedings of the National Academy of Sciences of the United States of America, 2001
- MMFF VI. MMFF94s option for energy minimization studiesJournal of Computational Chemistry, 1999
- Molecular basis of agonism and antagonism in the oestrogen receptorNature, 1997
- AIB1, a Steroid Receptor Coactivator Amplified in Breast and Ovarian CancerScience, 1997
- Identification of a new class of steroid hormone receptorsNature, 1988
- CHARMM: A program for macromolecular energy, minimization, and dynamics calculationsJournal of Computational Chemistry, 1983