Small-molecule FRET probes for protein kinase activity monitoring in living cells
- 9 July 2010
- journal article
- research article
- Published by Elsevier BV in Biochemical and Biophysical Research Communications
- Vol. 397 (4), 750-755
- https://doi.org/10.1016/j.bbrc.2010.06.026
Abstract
No abstract availableKeywords
Funding Information
- The Estonian Science Foundation (ETF8230)
- the EMES (SF0180121s08)
- the Fondation Leducq (O6 CVD 02)
- the NSF-NIH CRCNS program (NIH R01 AA18060)
- The British Heart Foundation (PG/07/091/23698)
This publication has 22 references indexed in Scilit:
- Adenosine analogue–oligo-arginine conjugates (ARCs) serve as high-affinity inhibitors and fluorescence probes of type I cGMP-dependent protein kinase (PKGIα)Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics, 2010
- The (un)targeted cancer kinomeNature Chemical Biology, 2010
- Structural Analysis of ARC-Type Inhibitor (ARC-1034) Binding to Protein Kinase A Catalytic Subunit and Rational Design of Bisubstrate Analogue Inhibitors of Basophilic Protein KinasesJournal of Medicinal Chemistry, 2008
- High-affinity bisubstrate probe for fluorescence anisotropy binding/displacement assays with protein kinases PKA and ROCKAnalytical Biochemistry, 2008
- High-Content Analysis of Kinase Activity in CellsCombinatorial Chemistry & High Throughput Screening, 2008
- Methodological and cellular aspects that govern the internalization mechanisms of arginine-rich cell-penetrating peptidesAdvanced Drug Delivery Reviews, 2007
- Surface-plasmon-resonance-based biosensor with immobilized bisubstrate analog inhibitor for the determination of affinities of ATP- and protein-competitive ligands of cAMP-dependent protein kinaseAnalytical Biochemistry, 2007
- Reading Dynamic Kinase Activity in Living Cells for High-Throughput ScreeningACS Chemical Biology, 2006
- Protein kinases — the major drug targets of the twenty-first century?Nature Reviews Drug Discovery, 2002
- Zwischenmolekulare Energiewanderung und FluoreszenzAnnalen der Physik, 1948