Bergaptol, a mechanism-based inactivator of CYP2C9
- 26 May 2020
- journal article
- research article
- Published by Springer Science and Business Media LLC in Medicinal Chemistry Research
- Vol. 29 (7), 1-8
- https://doi.org/10.1007/s00044-020-02564-x
Abstract
No abstract availableKeywords
Funding Information
- National Natural Science Foundation of China (81960754)
This publication has 19 references indexed in Scilit:
- Psoralen, a mechanism-based inactivator of CYP2B6Chemico-Biological Interactions, 2015
- Mechanism-based inactivation of cytochrome P450 2B6 by isopsoralenXenobiotica, 2015
- Mechanism-based inactivation of CYP450 enzymes: a case study of lapatinibDrug Metabolism Reviews, 2015
- Consumption of Clarified Grapefruit Juice Ameliorates High-Fat Diet Induced Insulin Resistance and Weight Gain in MicePLOS ONE, 2014
- Identification of the Residue in Human CYP3A4 That Is Covalently Modified by Bergamottin and the Reactive Intermediate That Contributes to the Grapefruit Juice EffectDrug Metabolism and Disposition, 2012
- Mechanism-Based Inactivation of Cytochrome P450 2C9 by Tienilic Acid and (±)-Suprofen: A Comparison of Kinetics and Probe Substrate SelectionDrug Metabolism and Disposition, 2008
- Potent Inhibition of Human Cytochrome P450 3A4, 2D6, and 2C9 Isoenzymes by Grapefruit Juice and Its FurocoumarinsJournal of Food Science, 2007
- Biosynthesis of coumarins in plants: a major pathway still to be unravelled for cytochrome P450 enzymesPhytochemistry Reviews, 2006
- Evidence-based drug–herbal interactionsLife Sciences, 2006
- Thiophene derivatives as new mechanism-based inhibitors of cytochromes P-450: Inactivation of yeast-expressed human liver cytochrome P-450 2C9 by tienilic acidBiochemistry, 1994